Literature detail

PPP2R5B regulates ANPEP expression and TGEV entry via dephosphorylation of HSF1 at Ser304/Ser308.

Yichen Yang1,2 Zhelin Su1,2 Xiyue Zhang1,2 Yubei Tan1,2 Hakimeh Baghaei Daemi1,2 Zhen Fu1,2 Meijie Gao1,2 Shengsong Xie3 Limeng Sun1,2 Guiqing Peng1,2,4,5
Affiliations 5 institutions
  1. State Key Laboratory of Agricultural Microbiology, College of Veterinary Medicine, Huazhong Agricultural University, Wuhan, China.
  2. Key Laboratory of Preventive Veterinary Medicine in Hubei Province, the Cooperative Innovation Center for Sustainable Pig Production, Wuhan, China.
  3. Key Laboratory of Agricultural Animal Genetics, Breeding and Reproduction of Ministry of Education & Key Lab of Swine Genetics and Breeding of Ministry of Agriculture and Rural Affairs, Huazhong Agricultural University, Wuhan, China.
  4. Key Laboratory of Prevention & Control for African Swine Fever and Other Major Pig Diseases, Ministry of Agriculture and Rural Affairs, Wuhan, China.
  5. Hubei Hongshan Laboratory, Frontiers Science Center for Animal Breeding and Sustainable Production, Wuhan, China.
PMID 42274214 2026 J Virol eng aheadofprint
PubMed DOI Browse context

Article

Publication summary

Transmissible gastroenteritis virus (TGEV) is an enteric coronavirus responsible for severe gastrointestinal disease in swine; however, the host determinants and mechanisms underlying viral entry remain poorly defined. This study systematically examines the role of the serine/threonine protein phosphatase 2A (PP2A) regulatory subunit B'β (PPP2R5B) during TGEV infection. Genetic ablation of PPP2R5B in PK-15 cells significantly reduced TGEV infectivity. Stage-specific analyses revealed that loss of PPP2R5B selectively impaired viral entry, while viral replication and release were unaffected. Transcriptomic profiling and functional validation identified the TGEV receptor aminopeptidase N (ANPEP) as a critical downstream effector of PPP2R5B. PPP2R5B-mediated regulation of ANPEP expression was independent of the AMPK, PI3K/AKT, ERK, and WNT/β-catenin signaling pathways. Instead, PPP2R5B directly interacted with heat shock factor 1 (HSF1) and promoted dephosphorylation of HSF1 at Ser304 and Ser308, thereby reducing HSF1-dependent transcriptional activation of ANPEP. These findings reveal a previously unrecognized PPP2R5B-HSF1-ANPEP regulatory axis that governs TGEV cellular entry and suggest that host dephosphorylation-dependent regulation may represent a potential target for antiviral intervention.IMPORTANCECoronavirus entry is a critical determinant of viral tropism and pathogenicity. This study identifies PPP2R5B, a regulatory subunit of the PP2A phosphatase complex, as a host factor that facilitates TGEV entry by controlling the expression of the cellular receptor ANPEP. We demonstrate that PPP2R5B regulates ANPEP transcription through modulation of HSF1 phosphorylation, independent of several canonical signaling pathways. These findings uncover a host phosphatase-dependent regulatory mechanism underlying coronavirus entry and highlight host signaling components as potential targets for antiviral intervention.

ANPEP coronavirus entry dephosphorylation HSF1 PPP2R5B

Structured evidence records

Evidence records

1 total
1 records
Extraction confidence 0.95
Key finding

PPP2R5B promotes transmissible gastroenteritis virus entry into PK-15 cells by dephosphorylating HSF1 at Ser304/Ser308, which enhances ANPEP receptor expression.

Virus
Host
Location
Not specified
Supporting text

Genetic ablation of PPP2R5B in PK-15 cells significantly reduced TGEV infectivity... PPP2R5B directly interacted with heat shock factor 1 (HSF1) and promoted dephosphorylation of HSF1 at Ser304 and Ser308, thereby reducing HSF1-dependent transcriptional activation of ANPEP.

Method
genetic ablation | transcriptomic profiling | functional validation
Sample type
PK-15 cells
Study design
in vitro experiment
Transmission direction
molecular mechanism only
Event type
host-factor regulation of receptor expression
Genes or proteins
PPP2R5B | ANPEP | HSF1
Receptors
ANPEP
Host factors
PPP2R5B | HSF1
Mutations
Ser304 | Ser308
Mechanism types
dephosphorylation-dependent receptor regulation